Dabrafenib

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Product Description

Dabrafenib is a compound used as a serine/threonine-protein kinase B-Raf inhibitor for oncology research. It competitively inhibits V600E BRAF gene mutations which are characteristic in melanoma cancers. Inhibition of B-Raf proteins, by dabrafenib, interrupts mitogen-activated protein kinase/extracellular signal regulated kinase (MAPK/ERK) pathways, which regulate cell growth.This action halts cell proliferative activity and engages apoptosis.

Product Specifications
Dabrafenib

Formula: C23H20F3N5O2S2

MW: 519.56 g/mol

Storage/Handling: Store desiccated at room temperature.

PubChem Chemical ID: 44462760

Product Specifications

Catalog ID D-210
CAS # 1195765-45-7
MW 519.56 g/mol

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